Apigenin (4',5,7-Trihydroxyflavone) is a competitive CYP2C9 inhibitor with a Ki of 2 μM. This natural flavonoid possesses broad biological properties including antioxidative, anti-inflammatory, anticancer, and neuroprotective effects.
- Competitive CYP2C9 inhibitor
- Exhibits antioxidative effects
- Exhibits anti-inflammatory effects
- Exhibits anticancer effects
- Exhibits neuroprotective effects
- Inhibits cell proliferation
- Alleviates Adriamycin (ADR)-induced myocardial injury